2020年
序号发表时间论文名称作者刊物、出版社名称卷、期(或章节)、页
12020-01Palladium-Catalyzed   Asymmetric [4+3] Cyclization of Trimethylenemethane: Regio-, Diastereo-, and   Enantioselective Construction of Benzofuro[3,2-b]azepine SkeletonsLiu   Yang-Zi, Wang Zhongao, Huang Zesheng, Zheng Xing, Yang Wu-Lin*, and Deng   Wei-Ping*Angew.   Chem. Int. Ed.2020, 59, 1238-1242
22020-07An   ArtemisininDerivative–(NHC)Gold(I)   Hybrid with Enhanced Cytotoxicity through Inhibition of NRF2 Transcriptional   ActivityChen   Zhang, Pierre-Yves Fortin, Guillaume Barnoin, Xue Qin  , Xing Wang, Alvaro Fernandez Alvarez,   Christian Bijani, Marie-Lise Maddelein, Catherine Hemmert*, Olivier   Cuvillier*  , Heinz Gornitzka*Angew.Chem.   Int. Ed.2020,   59, 12062-12068
32020-07Ribosomal   S6 protein kinase 4 promotes radioresistance in esophageal squamous cell   carcinoma.Mingyang   Li, Linni Fan, Donghui Han, Zhou Yu, Jing Ma, Yixiong Liu, Peifeng Li, Danhui   Zhao, Jia Chai, Lei Jiang, Shiliang Li, Juanjuan Xiao, Qiuhong Duan, Jing Ye,   Mei Shi, Yongzhan Nie, Kai-Chun Wu, Dezhong Joshua Liao, Yu Shi, Yan Wang,   Qingguo Yan, Shuangping Guo, Xiu-Wu Bian, Feng Zhu, Jian Zhang, Zhe Wang.J.   Clin. Invest.2020,   130(8), 4301-4319
42020-04A   single-component light sensor system allows highly tunable and direct   activation of gene expression in bacterial cellsXie   Li, Changcheng Zhang, Xiaopei Xu, Jun Miao, Jing Yao, Renmei Liu, Yuzheng   Zhao, Xianjun Chen,* and Yi Yang,*Nucleic   Acids Res.2020,   48(6), e33
52020-07Novel   and potent inhibitors targeting DHODH, a rate-limiting  enzyme in de novo pyrimidine biosynthesis,   are broad-spectrum antiviral against RNA viruses including newly emerged   coronavirus SARS-CoV-2Rui   Xiong, Leike Zhang, Shiliang Li, Yuan Sun, Minyi Ding, Yong Wang, Yongliang   Zhao, Yan Wu, Weijuan Shang, Xiaming Jiang, Jiwei Shan, Zihao Shen, Yi Tong,   Liuxin Xu, Yu Chen, Yingle Liu, Gang Zou, Dimitri Lavillete, Zhenjiang Zhao,   Rui Wang, Lili Zhu, Gengfu Xiao, Ke Lan, Honglin Li*, Ke Xu*Protein   Cell.2020, 11, 723–739
62020-04Illuminating   NAD(+) Metabolism in Live Cells and In Vivo Using a Genetically Encoded   Fluorescent SensorYejun   Zou, Aoxue Wang, Li Huang, Xudong Zhu, Qingxun Hu, Yinan Zhang, Xianjun   Chen,  Fengwen Li, Qiaohui Wang, Hu   Wang, Renmei Liu, Fangting Zuo, Ting Li, Jing Yao, Yajie Qian, Mei Shi, Xiao   Yue, Weicai Chen, Zhuo Zhang, Congrong Wang, Yong Zhou, Linyong Zhu, Zhenyu   Ju, Joseph Loscalzo, Yi Yang,* and Yuzheng Zhao*Dev.   Cell2020,   53, 1-13
72020-06First-generation   species-selective chemical probes for fluorescence imaging of human   senescence-associated β-galactosidase.Xiaokang   Li#, Wenjing Qiu#, Jinwen Li#, Xi Chen#, Yulu Hu, Ying Gao,   Donglei Shi, Xinming Li, Huiling Lin, Zelan Hu, Guoqiang Dong, Chunquan   Sheng, Bei Jiang, Conglong Xia, Chu-Young Kim, Yuan Guo*, Jian Li*.Chem.   Sci.2020,   11, 7292–7301
82020-05A   self-immobilizing near-infrared fluorogenic probe for sensitive imaging of   extracellular enzyme activity in vivoYuyao   Li, Heng Song, Chenghong Xue, Zhijun Fang, Liqin Xiong, and Hexin Xie*Chem.   Sci.2020,   11, 5889-5894
92020-01Targeting   virulence factors as an antimicrobial approach: Pigment inhibitors. Shuaishuai   Ni#, Baoli Li#, Yixiang Xu#, Fei Mao, Xiaokang Li,   Lefu Lan, Jin Zhu, Jian Li*.Med.   Res. Rev. 2020,   40, 293-338
102020-01Spatiotemporally   controllable diphtheria toxin
     expression using a light-switchable transgene system combining   multifunctional nanoparticle delivery system for targeted melanoma therapy
He,   Muye, Wang, Yan, Chen, Xianjun, Zhao, Yuzheng, Lou, Kaiyan, Wang, Yujie,   Huang, Lei, Hou, Xinyu, Xu, Jiajun, Cai, Xiaoran, Cheng, Yi, Lan, Minbo,   Yang, Yi*, Gao, Feng*J.   Control. Release2020, 319, 1-14
112020-05Lysosomal   polarity increases with aging as revealed by a lysosome-targetable   near-infrared fluorescent probe.Donglei   Shi#, Linghao Hu#, Xinming Li#, Wenwen Liu, Ying Gao,   Xiaokang Li, Bei Jiang, Conglong Xia, Yuan Guo*, Jian Li*.Sensor.   Actuator. B-Chem.2020,   319, 128302.
122020-10Sensitive   detection via the time-resolved fluorescence of circularly permuted yellow   fluorescent protein biosensorsLei   Li, Yuchi Cheng, Shiyu Shen, Jiasheng Zhou, Aoxue Wang, Guoqing Chen, Jianhua   Xua, Yi Yang, Yuzheng Zhao*, Sanjun Zhang*, Yang TianSensor.   Actuat. B-Chem.2020,   321, 128614
132020-3Repurposing   antimycotic ciclopirox olamine as a promising anti-ischemic stroke agent.Hongxuan   Feng#, Linghao Hu#, Hongwen Zhu#, Lingxue Tao#, Lei Wu, Qinyuan Zhao,   Yemi Gao, Qi Gong, Fei Mao, Xiaokang Li, Hu Zhou*, Jian Li*, Haiyan Zhang*.Acta   Pharm. Sin. B 2020,   10, 434–446
142020-1Discovery   of nitazoxanide-based derivatives as autophagy activators for the treatment   of Alzheimer's disease.Xiaokang   Li#, Jian Lu#, Yixiang Xu#, Jiaying Wang, Xiaoxia   Qiu, Lei Fan, Baoli Li, Wenwen Liu, Fei Mao, Jin Zhu, Xu Shen*, Jian Li*.Acta   Pharm. Sin. B 2020,   10, 646-666.
152020.04A   combination of LightOn gene expression system and tumor   microenvironment-responsive nanoparticle delivery system for targeted breast   cancer therapyXinyu   Hou, Chenting Shou, Muye He, Jiajun Xu, Yi Cheng, Zeting Yuan, Minbo Lan,   Yuzheng Zhao, Yi Yang, Xianjun Chen*, Feng Gao*Acta   Pharm. Sin. B 2020, 10(9),   1741-1753
162020-06Lighting   Up Live-Cell and In Vivo Central Carbon Metabolism with Genetically Encoded   Fluorescent SensorsZhuo   Zhang, Xiawei Cheng, Yuzheng Zhao*, and Yi Yang*Annu.   Rev. Anal. Chem.2020,   13(1), 293-314
172020.03Multiple   targeting strategies achieve novel protein drug deliver into cancer cells to   proapoptosis lung cancer cell by precisely inhibiting surviving. Fabiao   Hu,Ting Yan, Wei Guo, Qiuli Liu, Myong Hun Han, Chang Liu,Yuping Liu, Wenyun   Zheng*,  Fang You*, Yi Yang, Wenliang   Zhang and Xingyuan Ma*Nanoscale2020,   12, 10623-10638
18Oct-20Fluorophore-Promoted   Facile Deprotonation and Exocyclic Five-Membered Ring Cyclization for   Selective and Dynamic Tracking of Labile GlyoxalsHuan   Xu, Qianqian Liu, Xiaodong Song, Chao Wang, Xinru Wang, Shengnan Ma, Xiaolei   Wang, Yan Feng, Xiangming Meng, Xiaogang Liu,* Wei Wang,* and Kaiyan Lou*Anal.   Chem.2020,   92, 13829-13838
19Jul-05In   vivo Visualization of γ-Glutamyl transpeptidase Activity with an Activatable   Self-immobilizing Near-Infrared ProbeYuyao   Li, Chenghong Xue, Zhijun Fang, Weipan Xu, and Hexin Xie*Anal.   Chem.2020,   92, 15017-15024
202020-04Elaboration   of phosphoramidite ligands enabling palladiumcatalyzed diastereo- and   enantioselective all carbon [4+3] cycloadditionZheng   Xing, Sun Hao, Yang Wu-Lin*, Deng Wei-Ping*.Sci.   Chin. Chem.2020, 63, 911-916
212020-11Photodynamic   therapy induces autophagymediated cell death in human colorectal cancer cells   via activation of the ROS/JNK signaling pathwayChangfeng   Song, Wen Xu, Hongkun Wu, Xiaotong Wang, Qianyi Gong, Chang Liu, Jianwen Liu*   and Lin Zhou*Cell   Death Dis.2020,  11, 938-952
222020-02A   novel multistage antiplasmodial inhibitor targeting Plasmodium   falciparum histone deacetylase. Zhenghui   Huang#,*, Ruoxi Li#, Tongke Tang#, Dazheng Ling#, Manjiong Wang#, Dandan Xu#, Maoxin Sun, Lulu   Zheng, Feng Zhu, Hui Min, Rachasak Boonhok, Yan Ding, Yuhao Wen, Yicong Chen,   Xiaokang Li, Yuxi Chen, Taiping Liu, Jiping Han, Jun Miao, Qiang Fang, Yaming   Cao, Yun Tang, Jie Cui, Wenyue Xu, Liwang Cui, Jin Zhu, Gary Wong, Jian Li*,   Lubin Jiang*.Cell   Discov.2020,   6, 93
232020-05Identification   of the new covalent allosteric binding site of FBPase with disulfiram   derivatives toward glucose reduction.Yunyuan   Huang#, Yixiang Xu#, Rongrong Song#, Shuaishuai Ni#, Jiaqi Liu, Yanhong   Xu, Yanliang Ren*, Li Rao, Yingjie Wang, Lin Wei, Lingling Feng, Chen Su,   Chao Peng, Jian Li*, Jian Wan*.J.   Med. Chem.2020,   63, 6238–6247.
242020-01Development   of novel N-hydroxypyridone   derivatives as potential anti-ischemic stroke agentsLinghao   Hu#, Hong-Xuan   Feng#,   Hongguang Zhang, Songda Yu, Qinyuan Zhao, Wei Wang, Fengxia Bao, Xun Ding,   Jiajing Hu, Manjiong Wang, Yixiang Xu, Zengrui Wu, Xiaokang Li, Yun Tang, Fei   Mao*, Xiaoyan Chen, Haiyan Zhang*, Jian Li*.J.   Med. Chem.2020,   63, 1051-1067
252020-06Catalytic   Asymmetric [3+2] Annulation via Indolyl Copper-Allenylidene Intermediates:   Diastereo- and Enantioselective Assembly of Pyrrolo[-a]indolesZhang   Jian, Ni Tao, Yang Wu-Lin*, Deng Wei-Ping*Org.   Lett.2020, 22, 4547-4552
262020-05Organocatalytic   Regiodivergent Ring Expansion of Cyclobutanones for the Enantioselective   Synthesis of Azepino[ a]indoles and Cyclohepta[b]indolesYang   Wu-Lin*, Li Wen, Yang Zhong-Tao, Deng Wei-Ping*Org.   Lett.2020, 22, 4026-4032
272020-2Dimethylformamide-Modulated   Kdo Glycosylation for Stereoselective Synthesis of α‑Kdo Glycosides.Qixin   Lou, Qingting Hua, Liangliang Zhang, and You Yang*Org.   Lett.2020,   22(3), 981-985
282020-10Synthesis   of l-glycero- and d-glycero-d-manno-Heptose Building Blocks for   Stereoselective Assembly of the Lipopolysaccharide Core Trisaccharide of Vibrio parahemolyticus O2.Junchang   Wang, Jingjing Rong, Qixin Lou, Yirong Zhu, and You Yang*Org.   Lett.2020,   22(20), 8018-8022
292020-11Total   Synthesis and Immunological Evaluation of the Tri-d-glycero-d-manno-heptose   Antigen of the Lipopolysaccharide as a Vaccine Candidate against Helicobacter pylori.Junchang   Wang,§ Yiyue Zhang,§ Yirong Zhu, Junru Liu, Yan Chen, Xin Cao, and You Yang*Org.   Lett.2020,   22(22), 8780-8785
30Aug-20Enantioselective   [4 + 2] Cycloaddition Reaction of Vinylquinolines with Dienals Enabled by   Synergistic OrganocatalysisJing   Chen, Yiwei Fu, Yang Yu, Jian-Rong Wang, Yue-Wei Guo,* Hao Li,* and Wei Wang*Org.   Lett. 2020,   22, 6061-6066
312020-10Transition-Metal   Free Chemoselective Hydroxylation and Hydroxylation–Deuteration of   Heterobenzylic MethylenesYonghai   Liu, Yang Yu, Chengyu Sun, Yiwei Fu, Zhiguo Mang, Lei Shi, and Hao Li*Org.   Lett. 2020,   22, 8127–8131
32Jan-20A   cascade approach to 3D cyclic carbamates via an ionic decarboxylative   functionalization of olefinic oxamic acidsHuaqiang   Fan,‡ Yi Wan,‡ Peng Pan, Wenbin Cai, Shihui Liu, Chuanxu Liu* and Yongqiang   Zhang *Chem.   Commun.2020,   56, 86-89
332020-6Loss   of thioredoxin reductase function in a mouse stroke model disclosed by a   two-photon fluorescent probeJintao   Zhao, Yuan Qu, Hao Gao, Miao Zhong,    Xinming Li,  Fang Zhang, Yaxiong   Chen, Lu Gan,  Guodong Hu, Hong Zhang,  Shengxiang Zhang*  and    Jianguo Fang *Chem.   Commun.2020,56,   14075-14078
342020-2Structure-guided   engineering of Pseudomonas dacunhael-aspartate β-decarboxylase for   l-homophenylalanine synthesisMin   Zhang,  Pengfei Hu,  Yu-Cong Zheng,  Bu-Bing Zeng,   Qi Chen,    Zhi-Jun Zhang*  and  Jian-He Xu*  Chem.   Commun.2020,56,   13876-13879
35Jul-05A   novel method combining aptamer-Ag10NPs based microfluidic biochip with bright   field imaging for detection of KPC-2-expressing bacteriaJing   Chen, Hui Li, Hexin Xie*, Danke Xu*Anal.   Chim. Acta.2020,   113220-27
362020-10Kinetic   resolution of 2H-azirines via Cu(I)-catalyzed asymmetric 1,3-dipolar   cycloaddition of azomethine ylides.Deng   Hua, Liu Tian-Tian, Ding Zheng-Dong, Yang Wu-Lin, Luo Xiaoyan*, Deng   Wei-Ping*Org.   Chem. Front.2020, 7(20),   3247-3252
372020-3Copper(i)-catalyzed   asymmetric [3 + 3] annulation involving aziridines to construct   tetrahydro-β-carbolinesChao   Ye  Wu-Lin Yang, Yufei Zhai,  Hua   Deng,  Xiaoyan Luo*   Guoyin   Kai*  and  Wei-Ping DengOrg.   Chem. Front.2020,   7, 3393-3398
38Sep-20Graphitic   Carbon Nitride Polymer as a Recyclable Photoredox Catalyst for   Decarboxylative Alkynylation of Carboxylic AcidsJiaqi   Guo, Yating Wang, Yuhang Li, Kailin Lu, Shihui Liu, Wei Wang* and Yongqiang   Zhang,*Adv.   Synth. Catal.2020,   362, 2620-2625
39Jul-20Aldehydes   Switch Regioselectivity: a Prins Cyclization Strategy for the Synthesis of   Indoline-fused THFs and Indole-fused OxepanesXiaobei   Chen, Yuanrui Jiang, Huihui Geng, Xingyu Liu, Yizhuo Huang, Jingwei Lu,   Chenjing Gao, Shilei Zhang,* Jian Zhang,* and Wei Wang*Adv.   Synth. Catal.2020,   362, 2620 2625
402020-04Targeting   CD133 reverses drug-resistance via the AKT/NF-κB/MDR1 pathway in colorectal   cancer. Zeting   Yuan1, Xin Liang1, Yueping Zhan1, Ziyuan Wang, Jian Xu, Yanyan Qiu, Jie Wang,   Yijun Cao, Van-Minh Le, Hai-Trieu Ly, Jianhua Xu, Wei Li*, Peihao Yin*, Ke   Xu*. Br.   J. Cancer. 2020, 122(9),   1342-1353.
412020-7Development   of disulfide-derived fructose-1,6-bisphosphatase (FBPase) covalent inhibitors   for the treatment of type 2 diabetes.Yi-xiang   Xu#, Yun-yuan   Huang#,   Rong-rong Song#, Yan-liang Ren, Xin Chen, Chao Zhang, Fei Mao, Xiao-kang Li,   Jin Zhu, Shuai-shuai Ni*, Jian Wan*, Jian Li*. Eur. J. Med. Chem. 2020, 203, 112500
42Feb-20 Design, synthesis and evaluation of   diosgenin carbamate derivatives as multitarget anti-Alzheimer's disease   agentsGuixiang   Yang, Yan Huang, Lulu Zheng, Li Zhang, Lin Su, Yuhang Wu, Jie Li, Licheng   Zhou, Jin Huang, Yun Tang*, Rui Wang*, Lei Ma*Eur.   J. Med. Chem.2020,   187, 111913
432020-05Mesenchymal   stem cells combined with Liraglutide relieve acute lung injury through   apoptotic signaling restrained by PKA/β-catenin.Xiaotong   Yang, Xiaoying Ma, Ocholi Don, Yuanlin Song, Xiaoyan Chen, Jianwen Liu*,   Jieming Qu* and Yun Feng*Stem   Cell Res. Ther.2020, 11, 182-198
442020-2A   Novel Drug Delivery Carrier Comprised of Nimodipine Drug Solution and a   Nanoemulsion: Preparation, Characterization, in vitro, and in vivo StudiesSaixu   Huang,# Zhiyong Huang,# Zhiqin Fu,# Yamin Shi,, Qi   Dai, Shuyan Tang, Yongwei Gu, Youfa Xu, Jianming   Chen,, Xin Wu, and Fuzheng Ren*Int.   J. Nanomed.
2020,   15, 1161-1172
452020-01In silico prediction of binding   capacity and interaction forces of organic compounds with alpha- and   beta-cyclodextrinsPeiwen   Di, Jianhui Chen, Liping Liu, Weihua Li, Yun Tang*, Guixia Liu*J.   Mol. Liq.2020,   302, 112585
462020-01Discovery   and biological evaluation of   N-(3-(7-((2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)amino)-4-methyl-2-oxo-2H-pyrimido[4,5-d][1,3]oxazin-1(4H)-yl)phenyl)acrylamide   as potent Bruton’s tyrosine kinase inhibitorsMeng-zhen   Lai, Pei-ran Song, Dou Dou, Yan-yan Diao, Lin-jiang Tong, Tao Zhang, Hua   Xie*, Hong-lin Li*, Jian Ding*Acta   Pharmacol. Sin.2020, 41, 415-422
472020-04Natural   Product Piperine Alleviates Experimental Allergic Encephalomyelitis in Mice   by Targeting Dihydroorotate DehydrogenaseZehui   Liu, Qian Hu1,Wanyan Wang, Sisi Lu, Dang Wu, Shuyin Ze,
     Jiacheng He, Ying Huang, Wuyan Chen, Yechun Xu,Weiqiang Lu*, Jin
     Huang*
Biochem.   Pharmacol.2020,   177, 114000
482020-2Mechanistic   Insights into the Regio- and Stereoselectivities of Testosterone and   Dihydrotestosterone Hydroxylation Catalyzed
     by CYP3A4 and CYP19A1
Junhao   Li, Yun Tang, Weihua Li,* and Yaoquan Tu*Chem.   Eur. J. 2020, 26, 6214-6223
492020-08PTBP3   Induced Inhibition of Differentiation of Gastric Cancer Cells Through   Alternative Splicing of Id1. Bin   Chen, Weixia Chen, Xiaoyan Mu, Liyan Yang, Xiangyu Gu, Aiguang Zhao*, Xin   Liang*, Jianwen Liu*. Front.   Oncol. 2020, 10, 1477
502020-3Verapamil   extends lifespan in Caenorhabditis elegans by inhibiting calcineurin activity   and promoting autophagy.Wenwen   Liu#, Huiling Lin#, Zhifan Mao#, Lanxin Zhang, Keting   Bao, Bei Jiang, Conglong Xia, Wenjun Li, Zelan Hu*, Jian Li*.Aging-US 2020, 12, 5300–5317
512020-05Diastereoselective   Synthesis of Functionalized Tetrahydro-γ-Carbolines via a [3+3] Cycloaddition   of 2,2'-Diester Aziridines with β-(Indol-2-yl)-α,β-unsaturated KetonesZou   Xuejie, Liu Yangzi, Shang Shaojing, Yang Wulin*, Deng Wei-Ping*Chin.   Chem. Lett.2020, 31, 1293-1296
522020-1Discovery   of synergistic activity of fluoroquinolones in combination with antimicrobial   peptides against clinical polymyxin-resistant Pseudomonas   aeruginosa DK2.Xinyu   Zheng, Qiao Cao, Qin Cao, Fei Mao, Xiaokang Li, Jin Zhu*, Lefu Lan*, Jian Li*.Chin.   Chem. Lett. 2020,   31, 413–417
532020-6A   rapid-response near-infrared fluorescent probe with a large Stokes shift for   senescence-associated β-alactosidase activity detection and imaging of   senescent cells.Wenjing   Qiu#, Xiaokang Li#, Donglei Shi, Xinming   Li, Ying Gao, Jinwen Li, Fei Mao, Yuan Guo, Jian Li*.Dyes   Pigments2020,   182, 108657
542020-2Curcumin-based   polarity fluorescent probes: Design strategy and biological applications.Linghao   Hu#, Donglei Shi#, Xinming Li#, Jin Zhu, Fei Mao,   Xiaokang Li, Conglong Xia, Bei Jiang, Yuan Guo*, Jian Li*.Dyes   Pigments 2020, 177, 108320
552020-02Discovery   of a natural fluorescent probe targeting the Plasmodium falciparum cysteine   protease falcipain-2Lili   Zhu, Lei Shan, Junsheng Zhu, Li Li, Shiliang Li, Liyan Wang, Jiawei Wang,   Shoude Zhang, Hongchang Zhou, Weidong Zhang*, Honglin Li*Sci.   China Life Sci.2020, 63(7),   1016-1025
562020-06Computational   insights into molecular activation and positive cooperative mechanisms of   FFAR1 modulatorsDan   Teng, Jianhui Chen, Dongping Li, Zengrui Wu, Weihua Li, Yun Tang*, Guixia   Liu*J.   Chem. Inf. Model.2020,   60, 3214-3230
572020-08NetInfer:   a web server for prediction of targets, therapeutic and adverse effects via   network-based inference methods.Zengrui   Wu, Yayuan Peng, Zhuohang Yu, Weihua Li, Guixia Liu, and Yun Tang*J. Chem. Inf. Model.2020, 60(8),   3687-3691
582020-8Dissecting   the Structural Plasticity and Dynamics of Cytochrome P450 2B4 by Molecular   Dynamics SimulationsJunhao   Li, Yang Zhou, Yun Tang, Weihua Li,* and Yaoquan Tu*J.   Chem. Inf. Model. 2020,   60, 5026-5035
592020-2Computational   Insight into the Allosteric Activation Mechanism of Farnesoid X ReceptorYue   Chen, Junhao Li, Zengrui Wu, Guixia Liu, Honglin Li, Yun Tang,* and Weihua   Li*J.   Chem. Inf. Model. 2020,   60, 1540-1550
602020-4Copper   Promoted Aerobic Oxidative C(sp3)–C(sp3) Bond Cleavage of   N-(2-(Pyridin-2-yl)-ethyl)anilines Yang Yu, Yong Zhang, Chengyu Sun, Lei Shi,   Wei Wang*, and Hao Li*J.   Org. Chem. 2020,   85, 2725-2732
612020.01Safe   and Efficacious Diphtheria Toxin-Based Treatment for Melanoma: Combination of   a Light-On Gene-Expression System and NanotechnologyXu,   Jiajun, He, Muye, Hou, Xinyu, Wang, Yan, Shou, Chenting, Cai, Xiaoran, Yuan,   Zeting, Yin, Yu, Lan, Minbo, Lou, Kaiyan, Zhao, Yuzheng, Yang, Yi, Chen,   Xianjun*, Gao, Feng*Mol.   Pharmaceut.2020, 17(1), 301-315
622020-01Deep   Learning Based Drug Metabolites Prediction.Disha   Wang, Wenjun Liu, Zihao Shen, Lei Jiang, Jie Wang, Shiliang Li*, Honglin Li*Front.   Pharmacol.2020, 10, 1586
632020-4Drug–Drug   Cocrystals Provide Significant Improvements of Drug Properties in Treatment   with ProgesteroneChunyang   Guo, Qi Zhang, Bingqing Zhu, Zaiyong Zhang, Xiaoyu Ma, Wenjuan Dai, Xiaoyi   Gong, Guobin Ren*, and Xuefeng Mei*Cryst.   Growth Des. 2020,   20, 3053-3063
642020-10Pharmaceutical   Cocrystals of Nicorandil with Enhanced Chemical Stability and Sustained   ReleaseChunyang   Guo, Qi Zhang, Bingqing Zhu, Zaiyong Zhang, Junjie Bao, Qiaoce Ding, Guobin   Ren*, and Xuefeng Mei*Cryst.   Growth Des. 2020,   20, 6995-7005
652020-10Strategy   for efficient discovery of cocrystals via a network-based recommendation   model.Lulu   Zheng,# Bin Zhu,# Zengrui Wu, Xiaoxue Fang, Minghuang Hong, Guixia Liu,   Weihua Li, Guobin Ren,* and Yun Tang*Cryst. Growth   Des. 2020, 20(10),   6820-6830.
662020-07Shikonin   is a novel and selective IMPDH2 inhibitor that target triple-negative breast   cancerWanyan   Wang, YuWu, Si Chen, Xi Liu, Jiacheng He, Shuyi Wang, Weiqiang Lu*, Yong   Tang*, Jin Huang*Phytother.   Res.2020,   35(1), 463-476
672020-6Quercetin   inhibits virulence properties of Porphyromas gingivalis in periodontal   diseaseZhiyan   He, Xu Zhang, Zhongchen Song, Lu Li, Haishuang Chang, Shiliang Li* & Wei   Zhou*Scientifc   Reports2020,   10, 18313
682020-09 Highly Regio-, Diastereo-, and   Enantioselective Assembly of Azepino[2,3 b]indoles via Palladium-Catalyzed   [4+3] Cycloaddition.Yang   Wu-Lin, Huang Zesheng, Liu Yang-Zi, Yu Xingxin*, Deng Wei-Ping*Chin.   J. Chem.2020, 38(12),   1571-1574.
692020-05Catalytic   Enantioselective Formal Synthesis of MDM2 Antagonist RG7388 and Its AnalogueZou   Xue-Jie, Yang Wu-Lin*, Zhu Jing-Yan, Deng Wei-Ping*Chin.   J. Chem.2020, 38(5), 435-438
702020-09Insights   into the interaction mechanisms of estrogen-related receptor alpha (ERR   alpha) with ligands via molecular dynamics simulationsDongping   Li, Yingchun Cai, Dan Teng, Zengrui Wu, Weihua Li, Yun Tang*, Guxia Liu*J.   Biomol. Struct. Dyn.2020,   38, 3867-3878
712020-6Discovery   of novel and highly selective PI3Kδ inhibitors based on the p110δ crystal   structureWen-Qing   Jia,Ya-Ya Liu,Xiao-Yan Feng,Wei-Ren Xu &Xian-Chao Cheng*J.   Biomol. Struct. Dyn.2020,   38, 2499-2508
722020-2Virtual   identification of novel peroxisome proliferator-activated receptor (PPAR) α/δ   dual antagonist by 3D-QSAR, molecule docking, and molecule dynamics   simulationYa-Ya   Liu,Ting-Ting Ding,Xiao-Yan Feng,Wei-Ren Xu &Xian-Chao Cheng* J.   Biomol. Struct. Dyn.2020,   38, 4143-4161
732020-2Virtual   identification of novel PPARα/γ dual agonists by 3D-QSAR, molecule docking   and molecular dynamics studiesYa-Ya   Liu,Xiao-Yan Feng,Wen-Qing Jia,Zhi Jing,Wei-Ren Xu &Xian-Chao Cheng*J.   Biomol. Struct. Dyn.
2020,   38, 2672-2685
742020-8Characterization   and rational design for substrate specificity of a prolyl endopeptidase from   Stenotrophomonas maltophiliaJunjie   Yu, Junjie Wu, Dewei Xie, Lei Du, Ya-Jie Tang, Jingli Xie* Dongzhi Wei*Enzyme   Micro. Tech.2020,   138, 109548
75Jul-05A   minor structure modification serendipitously leads to a highly   carbapenemase-specific fluorogenic probeJie   Wang,‡ Weipan Xu,‡ Shuyuan Xue, Tao Yu and Hexin Xie*Org.   Biomol. Chem.2020,   18, 4029-4033
762020-10Synthesis   and Immunomodulatory Activity of the Sulfated Tetrasaccharide Motif of Type B   Ulvanobiuronic Acid 3-Sulfate.Liangliang   Zhang, Xiaotong Wang, Qingting Hua, Junchang Wang, Jianwen Liu* and You Yang*Org.   Biomol. Chem.2020,18(39), 7932-7935
772020-06The   immunosuppressant fingolimod ameliorates experimental autoimmune myasthenia   gravis by regulating T-cell balance and cytokine secretion.Yating   Luo, Yingfan Liang, Huan He, Mengting Zhang, Rui Wang*, Honglin Li*Am.   J Transl. Res.2020, 12(6),   2600-2613
782020-12Both   endogenous and exogenous miR-139-5p inhibit Fusobacterium nucleatum-related   colorectal cancer development.  Yuyu   Zhao, Qianying Tao, Shaoyu Li, Peiyong Zheng*, Jianwen Liu, Xin Liang*. Eur.   J. Pharmacol.2020, 888, 173459
792020-07A   Small-Scale Medication of Leflunomide as a Treatment of COVID-19 in an   Open-Label Blank-Controlled Clinical Trial.Ke   Hu, Mengmei Wang, Yang Zhao, Yunting Zhang, Tao Wang, Zhishui Zheng, Xiaochen   Li, Shaolin Zeng, Dong Zhao, Honglin Li*, Ke Xu*, Ke Lan*Virol.   Sin.2020, 35, 725-733
802020.04A   cytokine receptor domeless promotes white spot syndrome virus infection via   JAK/STAT signaling pathway in red claw crayfish Cherax quadricarinatus,  Ling-ke   Liu#, Xiao-xiao Chen#, Rui-lin Gaoa, Ke-jian Wanga, Wen-yun Zheng∗, Hai-peng   Liu∗Dev.   Comp. Immunol.2020,   111, 103749
812020-02In   silico prediction of human renal clearance of compounds using quantitative   structure-pharmacokinetic relationship modelsJianhui   Chen, Hongbin Yang, Lan Zhu, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*Chem.   Res. Toxicol.2020,   33, 640-650
822020-06Computational   approaches to identify structural alerts and their applications in   environmental toxicology and drug discoveryHongbin   Yang, Chaofeng Lou, Weihua Li, Guixia Liu, and Yun Tang*Chem. Res. Toxicol.2020, 33(6),   1312-1322
832020-03Hyperthermic   intraperitoneal chemotherapy with recombinant mutant human TNF and   raltitrexed in mice with colorectal-peritoneal carcinomatosis. Qianyi   Gong, Changfeng Song, Xiaotong Wang, Renjie Wang, Guoxiang Cai*, Xin Liang*,   Jianwen Liu*. Exp.   Biol. Med. (Maywood). 2020, 245(6), 542-551
842020-03Mesenchymal   stem cells maintain the stemness of colon cancer stem cells via   interleukin-8/mitogen-activated protein kinase signaling pathway. Xiaoying   Ma, Jiajun Liu, Xiaotong Yang, Kai Fang, Peiyong Zheng*, Xin Liang*, Jianwen   Liu*. Exp.   Biol. Med. (Maywood). 2020, 245(6),   562-575 
852020/9/1Facile   Preparation of 4‑(4-Nitrophenyl)morpholin-3-one via the Acid-Catalyzed   Selective Oxidation of 4‑(4-Nitrophenyl)morpholine by Sodium Chlorite as the   Sole OxidantChaoyang   Liu, Tao Yu, Tiannuo Yang, Haozhou Sun, Cheng Qin, Qiang Jia*, and Changhu   Chu*Org.   Process Res. Dev.2020, 24,   2633-2638 
862020-1Gastrointestinal   survival and potential bioactivities of Lactobacillus curieae CCTCC M2011381   in the fermentation of plant foodYafan   Liu, Yiji Zhang, Kum-Song Ro, Honglin Li, Lixin Wang, Jingli Xie*, Dongzhi   Wei*Process   Biochem. 2020, 88, 222-229
87Dec-20PIFA-Mediated   Cross-Dehydrogenative Coupling of N-Heteroarenes with Cyclic Ethers: Ethanol   as an Efficient PromoterXiang   Li+,Chaoyang Liu+, Shixun Guo, Wei Wang,* and Yongqiang Zhang*Eur.   J. Org. Chem. 2020,   1-12
882020-11Insights   into the mechanism of Arnebia euchroma on leukemia via network pharmacology   approach.Biting   Wang, Zengrui Wu*, Jiye Wang, Weihua Li, Guixia Liu, Bo Zhang and Yun Tang*BMC   Complem.Altern. M.2020, 20(1), 322
892020-03In   silico prediction of metabolic epoxidation for drug-like molecules via   machine learning methodsJiajing   Hu, Yingchun Cai, Weihua Li, Guixia Liu, and Yun Tang*Mol.   Inform.2020,   39(8), 1900178
90Sep-20Solubilization   of Hexyl Aminolevulinate by Surfactants for Tumor Fluorescence DetectionLirong   Ma, Xuanlin Yang, Xiuzhong Yao* and Weiyu Weng*Photochem.   Photobiol.2020,   96, 1088–1095
912020-2Facile   Construction of Troponoid Derivatives Incorporating Imidazolin-2-one MoietiesJing   Yu‡, Xiaobei Chen‡, Ye Liu, Bing Wu, Haiyan Li, Yanwei Hu∗, Liang Wang∗,   Shilei Zhang∗Synthesis-STUTTGART2020,   52(12), 1847-1854
922020-02Discovery   and optimization of 2-aminopyridine derivatives as novel and selective JAK2   inhibitorsXiangyu   Ma, Yanyan Diao, Huan Ge, Fangling Xu, Lili Zhu*, Zhenjiang Zhao*, Honglin   Li*Bioorg.   Med. Chem. Lett.2020, 30 (8), 127048
932020-06Design,   synthesis and biological evaluation of potent EGFR kinase inhibitors against   19D/T790M/C797S mutation.Zhicheng   Su, Tingyuan Yang, Jie Wang, Mengzhen Lai, Linjiang Tong, Gulinuer Wumaier,   Zhuo Chen*, Shengqing Li, Honglin Li, Hua Xie*, Zhenjiang Zhao*Bioorg.   Med. Chem. Lett.2020, 30(16), 127327
942020-5Repurposing   of antipsychotics perphenazine for the treatment of endometrial cancer. Yang   Chen#, Yunxia Cui#, Xiao Sun#, Huiwen Wu, Manjiao   Ou, Yunzhe Tang, Shuaishuai Ni, Xiaokang Li, Jin Zhu, Fei Mao*, Yudong Wang*,   Jian Li*.Bioorg.   Med. Chem. Lett. 2020,   30, 127239
95Dec-20Design,   synthesis and biological evaluation of novel osthole-based derivatives as   potential neuroprotective agentsLi   Zhang, Yuhang Wu, Guixiang Yang, Haixian Gan, Dayong Sang, Jiye Zhou, Lin Su,   Rui Wang*, Lei Ma*.Bioorg.   Med. Chem. Lett.2020,   30, 127633
962020-06In silico prediction of chemical   neurotoxicity using machine learningChangsheng   Jiang, Piaopiao Zhao, Weihua Li, Yun Tang*, Guixia Liu*Toxicol.   Res.2020,   9, 164-172
972020-10A   NaH-promoted N-detosylation reaction of diverse p-toluenesulfonamidesWanwan   Sun#, Xiaobei Chen#, Ying Hu, Huihui Geng, Yuanrui Jiang,   Yuxin Zhou, Wenjing Zhu, Min Hu, Haohua Hu, Xingyi Wang, Xinli Wang, Shilei   Zhang*, Yanwei Hu*Tetrahedron   Lett.2020,   61, 152442.
982020/12/1Activated   charcoal supported copper nanoparticles: A readily available and inexpensive   heterogeneous catalyst for the N-arylation of primary amides and lactams with   aryl iodidesRong   Zhao, Wenwen Dong, Jiangge Teng, Zhiwei Wang, Yunzhong Wang, Jianguo Yang,   Qiang Jia,  Changhu Chu*Tetrahedron 2020, 79, 131858
992020-6Design,   Synthesis and in Vitro Evaluation of Tylophorine Derivatives as Possible   Antitumor AgentsZhiguo   Mang  Shuai Zhang  Jing Bai    Meijuan Li  Hao Li*Chem.   Biodivers.2020,   17, e2000066
100Jul-20One-Pot   synthesis of isoindolin-1-ones with thiamine hydrochloride (VB1) as a   catalyst and their inhibitory activity against cancer cell lines.Pham   Van Khang, Lihong Hu, Lei Ma*.Polycycl.   Aromat. Comp. 2020, 40, 33-39
101Aug-20Dextran-based   Nanomicelle System with Directly Ester-bound Gadolinium Chelates as a   Magnetic Resonance Imaging Contrast Agent for Tumor Detection Lirong   Ma,1, Weiyu Yang,1, Dingmei Wu, Mengmeng Jiang, Xiuzhong Yao*and Weiyu Weng*Iran.   J. Pharm. Res.2020,   19 (3), 520-532
1022020.2聚乙烯亚胺改性的双介孔氧化硅基因载体构建方美蓉、   秦利梅、 贾晓博、 李永生、 牛德超*、 胡泽岚*无机材料学报2020, 35(2), 188-192
103May-20Design,   Synthesis and Biological Evaluation of Dimethyl Cardamonin (DMC) Derivatives   as P-glycoprotein-mediated Multidrug Resistance Reversal Agents. Ximeng   Shi, Yuyu Zhao, Licheng Zhou, Huanhuan Yin, Jianwen Liu*, Lei Ma*.Lett.   Drug Des. Discov.2020,   17, 1270-1282
1042020-5Identification   of Phosphoinositide-3 Kinases Delta and Gamma Dual Inhibitors Based on the   p110δ/γ Crystal StructureJia,   Wen-Qing; Feng, Xiao-Yan; Liu, Ya-Ya; Han, Zhen-Zhen; Jing, Zhi; Xu, Wei-Ren;   Cheng, Xian-Chao*Lett.   Drug Des. Discov.2020,   17, 772-786
1052020-2Study   on Drug Resistance to Tumor Cell in Oxygen Gradient and Co-culture   Microfluidic ChipSUN   Wei, CHEN Yu-Qing, WANG Ming-Fang, WANG Yue-Rong, ZHANG Min, ZHANG Hong-Yang,   HU Ping*Chinese   J. Anal. Chem.2020,   48(2), 180-186
106Jul-20Chemical   Compositions and Anti-cancer Activities of the Volatile Oils of Leaves and   Rhizomes of Three Polianthes Species.Pham   Van Khang*, Hoang Phu Hiep, Lei Ma, Sida Shen. Lett.   Org. Chem.2020,   17, 434-437
1072020-02Comparative   genomic analysis and proteolytic properties of Lactobacillus curieae CCTCC   M2011381Chen,   Y., Xie, J.*, Sun, J., Zhou, Z., Zhang, R., Li, H., Wei, DInt.   Food Res. J.2020, 27(5), 883-892
1082020-4Graphene   quantum dots in photodynamic therapyJiayi   Chen, Wentian Wu  Fangwei Zhang, Jiali Zhang, Hui   Liu, Jing Zheng*, Shouwu Guo* and Jingyan ZhangNanoscale   Adv.2020,   2, 4961-4967
1092020.3HZ-835大孔树脂分离甘草黄酮的研究韩伟、   姜文倩、 朱晓璐、 陈静雯徐州工程学院学报(自然科学版)2020, 35(01), 19-27
1102020-73-   脱氧-D - 甘露-2- 辛酮糖酸寡糖的合成研究进展庄丽琴,邓妤,曾铮,楼琦欣,杨友*药学进展2020, 44(7), 521-534
1112020-02靶向 PD-1 的多肽阻断剂的设计及评价全丽娜、刁妍妍、李巧、李文杰、朱丽丽、李洪林 华东理工大学学报(自然科学版)2020, 1, 35-40
1122020.1一种无孢灵芝菌丝体的活性成分岳亚文、   周帅、 冯杰、 王金艳、 唐庆九、 刘艳芳、 张劲松、 冯娜、 韩伟*菌物学报2020, 39(01), 128-136
1132020.1HPLC法测定灵芝孢子粉中三萜含量杨志空、   韩伟、 冯娜、 张劲松、 王晨光、 周靖、 王金艳*、 唐庆九*菌物学报2020,   39(01), 184-192
1142020.1高速逆流色谱法分离灵芝中的灵芝烯酸B岳亚文、   钱丁寅、 韩伟、 王晨光、 冯杰、 唐庆九、 张忠、 冯娜*、 张劲松*菌物学报2020,   39(01), 193-199
1152020.8灵芝菌丝体中一个三萜类化合物的核磁归属及活性初探朱晓璐、   岳亚文、 张劲松、 冯杰、 唐庆九、 冯娜、 韩伟*菌物学报2020,   39(08), 1551-1558
1162020.1灵芝孢子粉中脂溶性成分分析方法的建立杨志空、   王金艳、 冯娜、 张劲松、 王晨光、 严培兰、 周靖、 唐庆九、 韩伟*菌物学报2020,   39(10),  1971-1980
1172020.02蝉棒束孢菌孢梗束培植过程中主要成分含量的变化规律及其复方对小鼠睡眠的影响覃丽霞、王玉芹   、 李春如 、王静春、孙长胜、王春丽*菌物学报 2020, 39, 362-371
1182020.9吐温60协同微波提取甘草黄酮的优化姜文倩、   郑丹婷、 韩伟*南京工业大学学报(自然科学版)2020,   42(05),  671-676
1192020.9酒石酸亚铁-标准曲线法检测绿茶提取物中茶多酚含量邓祥、   韩伟*南京工业大学学报(自然科学版)2020,   42(05),  677-682
1202020-2羟基封端聚丁二烯的临界点色谱定量方法研究汪明芳、贾强强、王月荣、章弘扬、张敏、胡坪色谱 2020, 38(2), 238-243
1212020.1番石榴叶抑制酪氨酸酶作用机制研究 孙晓梦、林东明、杨弘、王禕、王凯晗、王春丽*食品研究与开发2020,   41(19), 64-68
1222020.06金露梅在酪氨酸酶催化中的抑制机理李晓雯、   王春丽*中成药2020,   42, 1585-1588


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